Compile Data Set for Download or QSAR
Found 19 of ic50 data for polymerid = 7374
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM12621(2,4-Diamino-5-ketopyrimidine 39 | 5-[(2,3-difluoro...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MPDPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50511926(CHEMBL4442620)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BM3PubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Inhibition of CDK3/Cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M94FZPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM454542(US10717746, Example 25 | US10717746, Example 84)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK3 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50528817(CHEMBL4462530 | US10717746, Example 14 | US2023041...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK3 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50511931(CHEMBL4579344)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of CDK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q21J2PubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)copy SMILEScopy InChI
Affinity DataIC50: 58nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MPDPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM454519(US10717746, Example 2)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of CDK3 (unknown origin) in presence of 5 mM ATPMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90D8VPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM164883(US9067888, 33)copy SMILEScopy InChI
Affinity DataIC50: 219nMpH: 7.5Assay Description:In vitro kinase assay analysis may be performed using standard techniques described in the art. These techniques are also used by commercial services...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CR5S4TUS Patent
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50601390(CHEMBL5177698)copy SMILES
Affinity DataIC50: 870nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5M3JPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50593922(CHEMBL5199065)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:Effective concentration required for inhibitory activity towards human beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50404389(CHEMBL5285499)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Effective concentration required for inhibitory activity towards human beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50267607(3-(5-Bromo-1-methyl-1H-indol-3-yl)-4-(6-hydroxymet...)copy SMILEScopy InChI
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of CDK3/Cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M94FZPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM164884(US9067888, 34)copy SMILEScopy InChI
Affinity DataIC50: 1.45E+3nMpH: 7.5Assay Description:In vitro kinase assay analysis may be performed using standard techniques described in the art. These techniques are also used by commercial services...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CR5S4TUS Patent
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50609501(CHEMBL5288241)copy SMILES
Affinity DataIC50: 1.84E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50434353(CHEMBL2386747 | US9446044, 72)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90DP7PubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50267760(3-Benzofuran-3-yl-4-(7-methoxymethyl-1-methyl-1H-i...)copy SMILEScopy InChI
Affinity DataIC50: 1.77E+4nMAssay Description:Inhibition of CDK3/Cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M94FZPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50267523(3-(6-Chloro-5-fluoro-1-methyl-1H-indol-3-yl)-4-(6-...)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of CDK3/Cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M94FZPubMed
TargetCyclin-dependent kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50267565(3-(6-Chloro-5-fluoro-1-methyl-1H-indol-3-yl)-4-(7-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK3/Cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24M94FZPubMed